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产地 | 中国 |
品牌 | Chemstan |
货号 | LC-01 |
用途 | 中间体 |
包装规格 | 20mg |
纯度 | 98%% |
CAS编号 | 1000413-72-8 |
是否进口 | 否 |
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Fields of Application :
TAK-875 is a potent, selective and orally bioavailable GPR40 agonist with EC50 of 0.072 μM.
CAS Number: | 1000413-72-8 |
Purity: | >98% |
Molecular Weight: | 524.63 |
Molecular Formula: | C29H32O7S |
Quality Control: HPLC、NMR、 LC/MS(Please contact us to get the QC report)
Synonyms: | TAK-875; TAK875; TAK 875. |
Chemical Name: | |
Storage: | 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO |
Note: Products for research use only, not for human use
Description:
TAK-875 is a potent, selective, and orally bioavailable GPR40 agonist, with a pharmacokinetic profile enabling long-acting drug efficacy. TAK-875 showed potent plasma glucose-lowering action and insulinotropic action during an oral glucose tolerance test in female Wistar fatty rats with impaired glucose tolerance. TAK-875 is currently in clinical trials For the treatment of type 2 diabetes mellitus.
References:
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