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产地 | 中国 |
品牌 | Chemstan |
货号 | CS-108742A |
用途 | 分析检测 |
包装规格 | 1mg |
纯度 | 99%% |
CAS编号 | |
是否进口 | 否 |
Description |
Abaloparatide TFA (BA 058 TFA) is a parathyroid hormone receptor 1 (PTHR1) analogue selected to be a potent and selective activator of the PTHR1 signaling pathway. Abaloparatide TFA enhances Gs/cAMP signaling (EC50 of 0.3 nM) and β-arrestin recruitment (EC50 of 0.9 nM) in MC3T3-E1 osteoblast cells[1] [2] . |
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IC50 & Target |
Parathyroid hormone receptor 1 (PTHR1) |
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