PD 168568 dihydrochloride-武汉科斯坦生物科技有限公司

产品展厅

您当前的位置：网站首页 > 产品展厅 >小分子化合物 >PD 168568 dihydrochloride

PD 168568 dihydrochloride

产品详请

产品描述
PD 168568 dihydrochloride is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).

体外活性
PD 168568 dihydrochloride has good selective for D4 receptor(Ki of 1842 nM for D2 receptor)[1].

体内活性
PD 168568 dihydrochloride inhibit amphetamine stimulated locomotor activity in the rat[1].

Cas No.
1782532-06-2

分子式
C22H29Cl2N3O

分子量

422.39

别名

PD 168568 (dihydrochloride);二盐酸PD168568

参考文献

[1]Belliotti TR, et al. Isoindolinone enantiomers having affinity for the dopamine D4 receptor. Bioorg Med Chem Lett. 1998 Jun 16;8(12):1499-502.

储存和溶解度
( < 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Note
For research use only .