PD 168568 dihydrochloride
- 价格： ￥382/支
- 发布日期： 2023-02-21
- 更新日期： 2025-05-13
产品详请
| 产地 |
China
|
| 品牌 |
TargetMol
|
| 货号 |
T12383
|
| 用途 |
Research Grade
|
| 包装规格 |
1mg
|
| 纯度 |
>98%%
|
| CAS编号 |
1782532-06-2
|
| 是否进口 |
否
|
产品描述
PD 168568 dihydrochloride is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).
体外活性
PD 168568 dihydrochloride has good selective for D4 receptor(Ki of 1842 nM for D2 receptor)[1].
体内活性
PD 168568 dihydrochloride inhibit amphetamine stimulated locomotor activity in the rat[1].
Cas No.
1782532-06-2
分子式
C22H29Cl2N3O
分子量
422.39
别名
PD 168568 (dihydrochloride);二盐酸PD168568
参考文献
[1]Belliotti TR, et al. Isoindolinone enantiomers having affinity for the dopamine D4 receptor. Bioorg Med Chem Lett. 1998 Jun 16;8(12):1499-502.
储存和溶解度
( < 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
Note
For research use only .
